About-cancer/treatment/drugs/breast

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Drugs Approved for Breast Cancer

This page lists cancer drugs approved by the Food and Drug Administration (FDA) for breast cancer. The list includes generic and brand names. This page also lists common drug combinations used in breast cancer. The individual drugs in the combinations are FDA-approved. However, the drug combinations themselves usually are not approved, although they are widely used.

The drug names link to NCI's Cancer Drug Information summaries. There may be drugs used in breast cancer that are not listed here.

Drugs Approved to Prevent Breast Cancer

Evista (Raloxifene Hydrochloride)

Raloxifene Hydrochloride

Tamoxifen Citrate

Drugs Approved to Treat Breast Cancer

Abemaciclib

Abraxane (Paclitaxel Albumin-stabilized Nanoparticle Formulation)

Ado-Trastuzumab Emtansine

Afinitor (Everolimus)

Afinitor Disperz (Everolimus)

Alpelisib

Anastrozole

Aredia (Pamidronate Disodium)

Arimidex (Anastrozole)

Aromasin (Exemestane)

Atezolizumab

Capecitabine

Cyclophosphamide

Docetaxel

Doxorubicin Hydrochloride

Ellence (Epirubicin Hydrochloride)

Epirubicin Hydrochloride

Eribulin Mesylate

Everolimus

Exemestane

5-FU (Fluorouracil Injection)

Fareston (Toremifene)

Faslodex (Fulvestrant)

Femara (Letrozole)

Fluorouracil Injection

Fulvestrant

Gemcitabine Hydrochloride

Gemzar (Gemcitabine Hydrochloride)

Goserelin Acetate

Halaven (Eribulin Mesylate)

Herceptin Hylecta (Trastuzumab and Hyaluronidase-oysk)

Herceptin (Trastuzumab)

Ibrance (Palbociclib)

Ixabepilone

Ixempra (Ixabepilone)

Kadcyla (Ado-Trastuzumab Emtansine)

Kisqali (Ribociclib)

Lapatinib Ditosylate

Letrozole

Lynparza (Olaparib)

Megestrol Acetate

Methotrexate

Neratinib Maleate

Nerlynx (Neratinib Maleate)

Olaparib

Paclitaxel

Paclitaxel Albumin-stabilized Nanoparticle Formulation

Palbociclib

Pamidronate Disodium

Perjeta (Pertuzumab)

Pertuzumab

Piqray (Alpelisib)

Ribociclib

Talazoparib Tosylate

Talzenna (Talazoparib Tosylate)

Tamoxifen Citrate

Taxol (Paclitaxel)

Taxotere (Docetaxel)

Tecentriq (Atezolizumab)

Thiotepa

Toremifene

Trastuzumab

Trastuzumab and Hyaluronidase-oysk

Trexall (Methotrexate)

Tykerb (Lapatinib Ditosylate)

Verzenio (Abemaciclib)

Vinblastine Sulfate

Xeloda (Capecitabine)

Zoladex (Goserelin Acetate)

Drug Combinations Used in Breast Cancer

AC

AC-T

CAF

CMF

FEC

TAC